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ML348
品牌:Badrilla
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ML348

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ML348

ML348

$60.00

In stock

Product code: A010-701
Unit Size: 1mg
  • Description
  • Data Sheet

ML348 is a competitive and reversible inhibitor of acyl palmitoyl thio-esterase 1 (APT1 – an enzyme encoded by the lysopholipase 1 gene (LYPLA1)). With a Ki = 300nM and an IC50 = 840nM, it exhibits a 14 fold greater selectivity for APT1 over APT2 (Ki and IC50 > 10µM).

Chemical name

N-[2-Chloro-5-(trifluoromethyl)phenyl]-4-(2-furanylcarbonyl)-1-piperazineacetamide

CAS number

899713-86-1

Molecular weight

415.79 g

Formula

C18H17ClF3N3O3

Solubility DMSO (48.5 mg/ml = 116.6 mM)
Purity ≥98%
Storage 4°C
Datasheet

A010-701

A010-701 MSDS

Regulatory statement Product for research use only. Not intended for diagnostic or therapeutic use.
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